找到约 2 条 “1191-85-1” 相关结果 (用时 0.375 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M20688 | B-Raf inhibitor 1 (Compound 13) dihydrochloride | B-Raf inhibitor 1 (Compound 13) dihydrochloride | Raf |
B-Raf inhibitor 1 (Compound 13) is a type IIA Raf inhibitor which bind to the DFG-out conformation with ki of 1 nM,1 nM,and 0.3 nM for B-Raf(WT), B-Raf(V600E) and C-Raf, respectively. | |||
M56345 | Eicosatetraynoic acid | Eicosatetraynoic acid | COX |
ETYA | |||
Eicosatetraynoic acid (ETYA) 是 cyclooxygenase 和 lipoxygenase 的非特异性抑制剂 (ID50=8 μM 和 4 μM)。Eicosatetraynoic acid (ETYA) 10 μM 激活 PPARα 和 PPARγ 嵌合体。 |