找到约 21 条 “AY77” 相关结果 (用时 0.109 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
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M3722
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Temsirolimus | 替西罗莫司;坦西莫司 | mTOR |
CCI-779; WAY-130779 | |||
Temsirolimus(WAY-130779,CCI-779)是一种mTOR的大环类抑制剂,在无细胞试验中IC50值为1.76 μM。 | |||
M7657 | Bay u9773 | Bay u9773 | Others |
Subtype-selective cysteinyl-leukotriene (Cys-Lt) antagonist. | |||
M14896
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Rogaratinib | Rogaratinib | FGFR |
BAY1163877 | |||
Rogaratinib (BAY1163877) 是一种有效且有选择性的成纤维细胞生长因子受体 (FGFR) 抑制剂。 | |||
M20047 | WAY-272077 | WAY-272077 | SPHK |
WAY-272077 is a haemostatic agent. | |||
M20053 | WAY-277054 | WAY-277054 | Others |
WAY-277054 is a tyrosine kinase inhibitor | |||
M20090 | WAY-320774 | WAY-320774 | Others |
WAY-320774 is a inhibitor of the Kanamycin Resistance Enzyme Eis from Mycobacterium tuberculosis | |||
M20148 | WAY-344977 | WAY-344977 | GSK-3 |
WAY-344977 is a inhibitor of Glycogen Synthase Kinase 3. | |||
M20169 | WAY-355772 | WAY-355772 | Serine/Threonine Protease |
WAY-355772 is a serine/threonine kinase inhibitor. | |||
M20202 | WAY-607738 | WAY-607738 | Others |
WAY-607738 is a inhibitor of Mcl-1 | |||
M20203 | WAY-607777 | WAY-607777 | Casein Kinase |
WAY-607777 is a Casein kinase 1d inhibitor. | |||
M20237 | WAY-633877 | WAY-633877 | Casein Kinase |
WAY-633877 is a Casein kinase 1δ inhibitor. | |||
M20262 | WAY-647729 | WAY-647729 | CDK |
WAY-647729 is a CDK9 inhibitor. | |||
M20263
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WAY-647766 | WAY-647766 | Casein Kinase |
Casein kinase 1δ-IN-4 | |||
WAY-647766是一种有效的 Casein kinase 1δ 抑制剂,可用于阿尔茨海默病的相关研究。 | |||
M20349 | WAY-311677 | WAY-311677 | FAK |
WAY-311677 is a novel anticancer agent (potential antiproliferation and FAK inhibitor). | |||
M20376 | WAY-277364 | WAY-277364 | Akt |
WAY-277364 is a Allosteric Akt inhibitor. | |||
M21909 | BAY-677 | BAY-677 | Others |
BAY-677 | |||
M27664 | BAY 60-2770 | BAY 60-2770 | Guanylate Cyclase |
BAY 60-2770 是一种有效的,选择性的,口服活性的可溶性鸟苷酸环化酶 (sGC) 活化剂。BAY 60-2770 以一氧化氮非依赖性方式增加 sGC 的活性。BAY 60-2770 具有抗纤维化作用。 | |||
M52910 | AY77 | AY77 | PAR |
AY77 是一种钙偏向的 PAR2 激动剂。 | |||
M58000 | CAY10770 | CAY10770 | Others |
CAY10770 | |||
M4505
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Sanggenone-D | 桑根酮D | Others |
Sanggenon D 是来自中国生药桑属 (Morus cathayana) 皮的 Diels-Alder 型加合物。 Sanggenon D 具有抗氧化作用,同时抑制胰脂肪酶 (PL),IC50 为 0.77 μM。 | |||
M52911 | AY254 | AY254 | PAR |
AY254 是 AY77 的类似物。 |