| M15983
|
6-Acetonyl-N-methyl-dihydrodecarine
|
6-Acetonyl-N-methyl-dihydrodecarine |
Alkaloids |
|
6-Acetonyl-N-methyl-dihydrodecarine |
| M15982
|
1-Methyl-2-pentyl-4(1H)-quinolinone
|
1-Methyl-2-pentyl-4(1H)-quinolinone |
Alkaloids |
|
1-Methyl-2-pentyl-4(1H)-quinolinone |
| M15981
|
1-Methyl-2-undecylquinolin-4(1H)-one
|
1-Methyl-2-undecylquinolin-4(1H)-one |
Alkaloids |
|
1-Methyl-2-undecylquinolin-4(1H)-one |
| M15980
|
3-Phenyl-1-(pyrrol-1-yl)propan-1-one
|
3-Phenyl-1-(pyrrol-1-yl)propan-1-one |
Alkaloids |
|
3-Phenyl-1-(pyrrol-1-yl)propan-1-one |
| M15979
|
7-Hydroxy-1-methoxy-3-methylcarbazole
|
7-Hydroxy-1-methoxy-3-methylcarbazole |
Alkaloids |
|
7-Hydroxy-1-methoxy-3-methylcarbazole |
| M15977
|
3,6-Dibenzyl-2-hydroxy-5-methoxypyrazine
|
3,6-Dibenzyl-2-hydroxy-5-methoxypyrazine |
Alkaloids |
|
3,6-Dibenzyl-2-hydroxy-5-methoxypyrazine |
| M15976
|
1,2-Dimethylquinolin-4-one-3-carboxylic acid
|
1,2-Dimethylquinolin-4-one-3-carboxylic acid |
Alkaloids |
|
1,2-Dimethylquinolin-4-one-3-carboxylic acid |
| M15975
|
6-Formyl-1,2,9,10-
tetramethoxy-6a,7-dehydroaporphine
|
6-Formyl-1,2,9,10-
tetramethoxy-6a,7-dehydroaporphine |
Alkaloids |
|
6-Formyl-1,2,9,10-
tetramethoxy-6a,7-dehydroaporphine |
| M15974
|
Indole-3-carboxylic acid
β-D-glucopyranosyl ester
|
Indole-3-carboxylic acid
β-D-glucopyranosyl ester |
Alkaloids |
|
Indole-3-carboxylic acid
β-D-glucopyranosyl ester |
| M8124
|
Quinine hemisulfate salt monohydrate
|
奎宁半硫酸盐一水合物 |
Potassium Channel |
|
Quinine hemisulfate salt monohydrate是一种钾离子通道 (potassium channel) 抑制剂,可抑制电压脉冲引起的 MT mSlo3 (KCa5.1) 通道 +100 mV 电流, 其 IC50 值为 169 μM。此外,Quinine hemisulfate salt monohydrate还能以低纳摩尔亲和力与嘌呤核苷磷酸化酶(PfPNP)结合。 |
| M7647
|
Bryostatin 1
|
苔藓抑素1 |
PKC |
|
Bryostatin 1是一种从苔藓虫 Bugula neritina 中分离出来的天然大环内酯类化合物,同时也是有效的中枢神经系统 (CNS) 渗透性的 PKC 调节剂。Bryostatin 1 能以 Ki 值为 8.07 nM 和 0.45 nM 分别结合到分离的 Munc13-1 的 C1 域和全长的 Munc13-1 蛋白,并具有抗癌,抗炎以及神经保护活性。 |